2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.
-
date post
19-Dec-2015 -
Category
Documents
-
view
218 -
download
2
Transcript of 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.
![Page 1: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/1.jpg)
2003-2004CNS Pharmacology
Review
April 18, 202308:30 PM
![Page 2: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/2.jpg)
Acetaminophen
Analgesic, Antipyretic
![Page 3: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/3.jpg)
Adrenocorticotropin(ACTH)
Anterior pituitary hormoneAnticonvulsant
Stimulates synthesisand release of cortisol
![Page 4: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/4.jpg)
Alfentanil
OpioidGeneral anaesthetic
Intravenous anaesthetic
![Page 5: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/5.jpg)
Amantadine
AntiviralAntiparkinson
Treatment of Influenza A Inhibits replication
at the stage of uncoatingInhibits dopamine release
![Page 6: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/6.jpg)
Amitriptyline
Tricyclic antidepressant (TCA)
![Page 7: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/7.jpg)
Amphetamine
Indirect sympathomimeticDrug of abuse
ADD treatmentStimulant
![Page 8: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/8.jpg)
Atropine
Anticholinergic
AntimuscarinicTreatment for bradycardia,
diarrhea, cholinesterase poisoning
![Page 9: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/9.jpg)
Baclofen
Skeletal muscle relaxantAnxiolytic
GABAB agonist
![Page 10: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/10.jpg)
Benztropine
AnticholinergicAntiparkinson
Muscarinic receptor antagonist
![Page 11: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/11.jpg)
Bethanecol
Cholinomimetic
Muscarinic agonistInduces defecation and
urinationBronchoconstrictor
![Page 12: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/12.jpg)
Bromocriptine
Antiparkinson
Dopamine (D2) agonistInhibits prolactin release
![Page 13: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/13.jpg)
Brupropion
Second generation antidepressant
![Page 14: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/14.jpg)
Buprenorphine
Opioid
Partial agonist
![Page 15: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/15.jpg)
Buspirone
Sedative/hypnoticAnxiolytic
![Page 16: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/16.jpg)
Butorphanol
OpioidAnalgesic
receptor partial agonistor antagonist
![Page 17: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/17.jpg)
Carbamazepine
Anticonvulsant
![Page 18: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/18.jpg)
Carbidopa
Antiparkinson
Peripheral dopa decarboxylase inhibitor
![Page 19: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/19.jpg)
Celecoxib
NSAIDAnti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
![Page 20: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/20.jpg)
Chloral hydrate
Sedative/HypnoticGeneral anaesthetic
Acts on GABAA receptor complexSimilar to barbiturates
![Page 21: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/21.jpg)
Chlordiazepoxide
Sedative/hypnoticAnxiolytic
Benodiazepine Acts on GABAA receptor
complex
![Page 22: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/22.jpg)
Chlorpromazine
Antipsychotic
Phenothiazine
![Page 23: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/23.jpg)
Clozapine
Antipsychotic
![Page 24: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/24.jpg)
Cocaine
Indirect sympathomimeticDrug of abuse
Topical anaesthetic
StimulantLocal anaesthetic
![Page 25: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/25.jpg)
Codeine
OpioidAnalgesic
Weak agonist
![Page 26: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/26.jpg)
Dantrolene
Skeletal muscle relaxant
Ryanodine receptor antagonistTreatment for malignant hyperthermia
![Page 27: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/27.jpg)
Deprenyl/selegiline
Antiparkinson
Monoamine oxidase B inhibitor(MAO-I)
Potentiates effects of L-Dopa
![Page 28: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/28.jpg)
Desipramine
Tricyclic antidepressant (TCA)
![Page 29: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/29.jpg)
Dextromethorphan
Opioid
Antitussive
![Page 30: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/30.jpg)
Diazepam
Sedative/hypnoticAnxiolytic
Anticonvulsant
Benzodiazepine Acts on GABAA receptor complex
![Page 31: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/31.jpg)
Diflunisal
NSAIDAnalgesic, Anti-inflammatory
Antipyretic
Cyclooxygenase inhibitor
![Page 32: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/32.jpg)
Diphenoxylate docusate
Antidiarrheal
Opiate
![Page 33: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/33.jpg)
Enflurane
General anaesthetic
Inhaled anaesthetic
![Page 34: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/34.jpg)
Entacapone
Antiparkinson
Peripheral catechol-o-methyltransferase inhibitor
![Page 35: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/35.jpg)
Ephedra(Ma Huang)
Dietary supplement
Amphetamine-like stimulant
![Page 36: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/36.jpg)
Ethanol
Drug of abuse
Sedative
![Page 37: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/37.jpg)
Ethosuximide
Anticonvulsant
![Page 38: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/38.jpg)
Etomidate
General anaesthetic
Intravenous anaesthetic
![Page 39: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/39.jpg)
Fentanyl
OpioidAnalgesic
receptor agonist
![Page 40: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/40.jpg)
Flumazenil
Benzodiazepine antagonist
Acts on GABAA receptor complex
![Page 41: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/41.jpg)
Fluoxetine
Antidepressant
Selective serotonin reuptake inhibitor (SSRI)
![Page 42: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/42.jpg)
Flurazepam
Sedative/Hypnotic
Benzodiazepine Acts on GABAA receptor
complex
![Page 43: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/43.jpg)
Ginko biloba
Dietary supplement
Treatment of Alzheimer symptoms
![Page 44: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/44.jpg)
Glutethimide
Sedative/Hypnotic
![Page 45: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/45.jpg)
Haloperidol
Antipsychotic
![Page 46: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/46.jpg)
Halothane
General anaesthetic
Inhaled anaesthetic
![Page 47: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/47.jpg)
Heroin
Drug of abuse
Opioid
![Page 48: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/48.jpg)
Imipramine
Indirect sympathomimeticTricyclic antidepressant (TCA)
Antimicturant
![Page 49: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/49.jpg)
Indomethacin
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitorTocolytic
Uterine relaxant
![Page 50: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/50.jpg)
Isoflurane
General anaesthetic
Inhaled anaesthetic
![Page 51: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/51.jpg)
Kava kava
Dietary supplement
Stress relief andtreatment of insomnia
![Page 52: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/52.jpg)
Ketamine
General anaestheticDrug of abuse
Sedative
![Page 53: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/53.jpg)
Ketoprofen
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
![Page 54: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/54.jpg)
Levodopa
Antiparkinson
Dopamine precursor
![Page 55: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/55.jpg)
Lidocaine
Class I antiarrhythmicLocal anaesthetic
Na+ channel blocker(activated and inactivated channels)
![Page 56: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/56.jpg)
Lithium
Antidepressant
Used to treatmanic/depressive disorder
![Page 57: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/57.jpg)
Loperamide
Antidiarrheal
Opiate
![Page 58: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/58.jpg)
Lorazepam
AnxiolyticAnticonvulsant
BenzodiazepineActs on GABAA receptor complex
![Page 59: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/59.jpg)
Lysergic acid diethylamide
(LSD)
Drug of abuse
Hallucinogen
![Page 60: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/60.jpg)
Marijuana
Drug of abuse
Cannabinoid
![Page 61: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/61.jpg)
Meperidine
Opioid analgesic
receptor agonist
![Page 62: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/62.jpg)
Mepivacaine
Local anaesthetic
![Page 63: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/63.jpg)
Meprobamate
Sedative/hypnoticAnxiolytic
![Page 64: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/64.jpg)
Meclofenamate
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
![Page 65: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/65.jpg)
Metamphetamine
Drug of abuse
Stimulant
![Page 66: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/66.jpg)
Methadone
Opioid
receptor agonist
![Page 67: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/67.jpg)
Morphine
OpioidAnalgesic
receptor agonist
![Page 68: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/68.jpg)
Nalbuphine
Opioid antagonist
receptor antagonist
![Page 69: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/69.jpg)
Nalmefene
Opioid antagonist
![Page 70: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/70.jpg)
Nalorphine
Opioid antagonist
![Page 71: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/71.jpg)
Naloxone
Opioid antagonist
![Page 72: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/72.jpg)
Naltrexone
Opioid antagonist
![Page 73: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/73.jpg)
Naproxen
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
![Page 74: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/74.jpg)
Neostigmine
Anticholinesterase
VasodilatorTreatment for myaesthenia gravisPromotes defecation and urination
Bronchoconstrictor
![Page 75: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/75.jpg)
Nicotine
CholinomimeticDrug of abuse
Nicotinic receptor agonist(skeletal muscle contraction)
StimulantSmoking cessation medication
![Page 76: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/76.jpg)
Nitrous oxide
General anaesthetic
Inhaled anaesthetic
![Page 77: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/77.jpg)
Non-steroidalAnti-inflammatory Drugs
(NSAIDs)
Analgesic, Anti-inflammatory, Antipyretic
Cyclooxygenase inhibitors
![Page 78: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/78.jpg)
Nortriptyline
Tricyclic antidepressant (TCA)
![Page 79: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/79.jpg)
Oxazepam
Sedative/hypnoticAnxiolytic
BenzodiazepineActs on GABAA receptor complex
![Page 80: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/80.jpg)
Oxybutinin
Anticholinergic
Muscarinic receptor antagonistPrevents urination
![Page 81: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/81.jpg)
Oxycodone
Analgesic
Opioid agonist
![Page 82: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/82.jpg)
Paraldehyde
Sedative/Hypnotic
![Page 83: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/83.jpg)
Pentazocine
Opioid analgesic
receptor partial agonist or antagonist
![Page 84: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/84.jpg)
Pentobarbital
Sedative/Hypnotic
Barbiturate
![Page 85: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/85.jpg)
Phencyclidine (PCP)
Drug of abuse
Hallucinogen
![Page 86: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/86.jpg)
Phenobarbital
Sedative/HypnoticAnticonvulsant
Barbiturate
![Page 87: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/87.jpg)
Phenytoin
AnticonvulsantClass I antiarrhythmic
Na+ channel blocker(inactivated channels)
![Page 88: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/88.jpg)
Piroxicam
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
![Page 89: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/89.jpg)
Pramipexole
Antiparkinson
Dopamine agonist (non-ergot)
![Page 90: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/90.jpg)
Primidone
Anticonvulsant
![Page 91: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/91.jpg)
Procaine
Local anaesthetic
![Page 92: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/92.jpg)
Propofol
General anaesthetic
Intravenous anaesthetic
![Page 93: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/93.jpg)
Resperidone
Antipsychotic
![Page 94: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/94.jpg)
Ropinirole
Antiparkinson
Dopamine agonist (non-ergot)
![Page 95: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/95.jpg)
Sertraline
Antidepressant
Selective serotonin reuptake inhibitor (SSRI)
![Page 96: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/96.jpg)
Sildenafil
Vasodilator
Promotes erection
![Page 97: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/97.jpg)
St. John’s Wort
Dietary supplement
Antidepressant
![Page 98: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/98.jpg)
Sufentanil
OpioidGeneral anaesthetic
Intravenous anaesthetic
![Page 99: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/99.jpg)
Sulindac
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
![Page 100: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/100.jpg)
Temazepam
Sedative/Hypnotic
BenzodiazepineActs on GABAA receptor complex
![Page 101: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/101.jpg)
Tetracaine
Local anaesthetic
![Page 102: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/102.jpg)
Thiopental
General anaesthetic
Ultra-short-acting barbiturate
![Page 103: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/103.jpg)
Thioridazine
Antipsychotic
Phenothiazine
![Page 104: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/104.jpg)
Thiothixene
Antipsychotic
![Page 105: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/105.jpg)
Tolterodine
Anticholinergic
Muscarinic receptor antagonistPrevents urination
![Page 106: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/106.jpg)
Tranylcypromine
Antidepressant
Monoamine oxidase inhibitor (MAO-I)
![Page 107: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/107.jpg)
Triazolam
Sedative/Hypnotic
BenzodiazepineActs on GABAA receptor complex
![Page 108: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/108.jpg)
Trifluoperazine
Antipsychotic
Phenothiazine
![Page 109: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/109.jpg)
Trihexyphenidyl
Antiparkinson
Antimuscarinic
![Page 110: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/110.jpg)
Valproic acid
Anticonvulsant
![Page 111: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/111.jpg)
Vigabatrin
Anticonvulsant
Irreversible GABA aminotransferase inhibitor
![Page 112: 2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM.](https://reader035.fdocuments.us/reader035/viewer/2022062421/56649d355503460f94a0d2e8/html5/thumbnails/112.jpg)
Zolpidem
Sedative/Hypnotic
Non-benzodiazepine