Understand the target first
Wi comment on Molecular Design.
Protein Pocket
a cat’s face
Let’s make analogy …
Inhibitor
Star Corps Trooper Helmet
Wi
Tom&Jerry
(Fluff) Syri
Garfield
Sylvester
Charmmy Kitty
Hello Kitty
Low resolution& Complex
Felix
Wi
Tom&Jerry
(Fluff) Syri
Garfield
Sylvester
Charmmy Kitty
Hello Kitty
Side effectsFelix
Wi
Tom&Jerry
(Fluff) Syri
Garfield
Sylvester
Charmmy Kitty
Hello Kitty
Multi-targeting
Felix
Wi
Tom&Jerry
(Fluff) Syri
Garfield
Sylvester
Charmmy Kitty
Hello Kitty
Specific
Felix
Wi
Tom&Jerry
(Fluff) Syri
Garfield
Sylvester
Charmmy Kitty
Hello Kitty
Felix
Wi
Doraemon
TargetDesign
For discussion, email me:
mbduangrudee@mahidol.ac.th