Contents of volume 16
Transcript of Contents of volume 16
CONTENTS OF VOLUME 16
Vol. 16, No. 1
Minireviews
Robert P. Hof
F. A. Wali
General Papers
Arun P. Kulkarni and Ileana Gonzales
J. W. Phillis
Godfrey Tunnicliff, Kathy L. Welborn and That T. Ngo
Hans Kriiger, Regina Gr~itz and Helga Grahn
M. Grau and J. Balasch
M. Alfonso, M. A. Parafita, M. J. Mancebo and J. Marc6
Unto Nousiainen
T. R. Hall, G. Uruefia and H. R. Figueroa
H. Meshkinpour, D. Hollander, D. Harmon and S. Koyama
M. L. Laorden, J. Hermindez and A. J. Brugger
L. Michaiska, G. Nagel, E. Swiniarski and M. M. Zydowo
Viviana Tarizzo and Modesto C. Rubio
13
19
25
31
37
43
PY 108-068: a calcium antagonist with an unusual pattern of cardiovascular activity
7 General anaesthetics: effects on transmitter release
49
55
61
65
69
Stimulation of the mouse hepatic microsomal aniline p- hydroxylases by acetone and polyamines
Chlorpromazine and trifluoperazine potentiate the action of adenosine on rat cerebral cortical neurons
Identification of potential GABA-mimetics by their actions on brain GABA recognition sites
Influence of ethanol upon the introduction of tyrosine amino- transferase in liver, upon the NAD content in liver and brain, and upon the activity of glutamate oxalate aminotransferase and glutamate pyruvate aminotransferase in the serum of rats
Protective effects of "cerebroactive drugs" in a model of acute hypoxia
Further evidence for effects of ethanol on gonadotrophins and prolactin secretion in female rats
Effects of phenobarbital and p , p ' - D D T on carboxylesterase activity and hydrolysis of propanidid in rat liver
Changes in mouse brain serotonin turnover following chronic imipramine administration
Colonic absorption of 1,2-dimethyl hydrazine (DMH) in the rat
The beta-agonist drug tulobuterol decreases cardiac auto- maticity in the rat: comparison with isoproterenol
The effect of ~-solanine on the active calcium transport in rat intestine
71 Effects of cocaine on several adrenergic system parameters
A. N. Elias, N. D. Vaziri, L. J. Deftos, R. Shinto and L. J. Valenta
75 Effect of bromocriptine on serum PTH, calcium and phos- phate levels in azotemic rats
New Patents i New patents and published patent applications from the United States and over 30 other countries
Minireview
lan Kitchen 79
Vol. 16, No. 2
Endogenous opioid nomenclature: light at the end of the tunnel
iii G P I~ 6,~H
General Papers Cheng S. Tsai and Richard F. Ochillo
Masahiro Aomine and Makoto Arita
George B. Weiss and Phyllis Kutsky
H. R. Figueroa, P. B. Yiirgens, D. K. Newton and T. R. Hall
G. Baifag6n, J. A. Arranz and E. J. Marco
G. liliano, R. Galderisi, A. Di Donato, G. Paofisso and G. F. Draetta
Ritsuko Matsukawa, Mitsuo Hayakawa, Minoru Tanaka and Hisashi Takiguchi
Yoshiaki Akimoto, Hitoshi Nishimura, Masamichi Komiya, Tomomi Shibata, Kenji Kaneko, Akira Fujii and Toyoyuki Tamura
A. Hellegouarch, J. Baran~s, F. Clostre, K. Drieu, P. Braquet and F. V. DeFeudis
Kiyoshi Sakai, Kuniko Higuchi-Nakamura and Masaatsu-Koujiro Uchida
K. F. A. Soliman and N. N. Gabriel
N. D. Vaziri, C. Byrne, C. H. Barton, D. Robertson, K. Jay and L. McDonald
C. A. Taira and M. A. Enero
Lilla Lachowicz and Gra~yna Janiszewska
Birger Kaada and Idar Lygren
Pedro Garz6n, Sonia Roman-Maidonado, Alicia Navarro-Ruiz and Pedro Solis-Camara V
Book Reviews
85
91
97
103
Comparative studies of cardiovascular effects of a new dopamine agonist (SK&F 38393A) and dopamine
Pretreatment with coenzyme Q,0 protects guinea pig ventric- ular muscle from hypoxia-induced deterioration of action potentials and contraction
Effects of manganese on 45Ca mobilization and contractile responses in rabbit aortic smooth muscle
Evidence for negative feedback control of the release of [3H]serotonin from superfused mouse cerebellum slices in- duced by electrical field stimulation
109 Indirect adrenergic effect of histamine in cat right atrium
115
121
125
129
133
137
141
145
149
153
The effects of lidocaine and procainamide on the sarco- lemmal membrane high affinity cyclic AMP phospho- diesterase of rat myocardium
Prostaglandin A 2 receptor in rat intestinal basolateral plasma membranes
Ampicillin concentrations in human serum, gingiva, the mandibular bone, and dental follicle following a single oral administration
Comparison of the contractile effects of an extract of Ginkgo biloba and some neurotransmitters on rabbit isolated vena cava
Calcium reversal: inhibition by Ca ion of sustained con- traction in Ca-free medium induced by various agonists in rat uterine smooth muscle
Brain cholinergic involvement in the rapid development of tolerance to the hypothermic action of ethanol
Prevention of metabolic alkalosis induced by gastric fluid loss using H 2 receptor antagonist
Participation of cholinergic pathways in sinoaortic de- nervated rats
Role of theophylline during the action of SP in vitro on the activity of synaptosomal membrane ATPase (EC 3,6.1.3) from different areas of rat brain
Lower plasma levels of some gastrointestinal peptides m Raynaud's disease. Influence of transcutaneous nerve stimulation
157 Response of rats to seizure stimulus modified by feeding
161
iv
Review Edward K. Y. Chiu and 163 J. Steven Richardson
General Papers Jun-lchi Nishijima, 177 Mitsuhiro Okamoto, Kazunori Nakaguchi, Michio Ogawa, Toshio Yamano and Takesada Mori
C. Giunta, M. De Bortoli, 183 M. Sanchini and A. Stacchini
Gregory A. Beumel and 189 Ernest Hodgson
Gregory A. Beumel, Patricia E. Levi 193 and Ernest Hodgson
Kazuhiko Ohishi, Tamiko Suzuki and Masaatsu K. Uchida
Clement Judes, Jean-Jacques Helwig, Claude Bollack and Paul Mandel
199
205
Jiann-Wu Wei and Der-Huey Chiang 211
Kohji Fujii, Ryuji Inoue, Kiyoichiroh Yamanaka and Takeshi Yoshitomi
217
Armand Lione 223
Jan I. M. Drayer, Michael A. Weber and Patricia P. Frankfort
229
A. O. Savage and G. K. Atanga 235
J. G. Auc~lio, J. B. Calixto and A. Jurkiewicz
J. Marin, C. Lazcano, L. Recio, M. Salaices and C. F. Sanchez-Ferrer
Steven G. Kamerling, David J. DeQuick, Timothy J. Weckman and Thomas Tobin
C. Cortinovis, D. Mayer, B. Bouscarel, H. Paris and J. C. Murat
I. Takayanagi and K. Koike
I. Takayanagi, K. Okumura and K. Koike
241
247
253
259
265
Vol. 16, No. 3
Behavioral and neurochemical aspects of prostaglandins in brain function
Inhibitory effect of gabexate mesilate on pancreatic phos- pholipase Az-mediated hydrolysis of ghost membranes
Activatory effect of two cardioglycosides on Cavia cobaya kidney Na+/K+-ATPase activity
The binding of isocyanides to cytochrome P-450 from mouse hepatic microsomes
Spectral interactions of piperonyl butoxide and isocyanides with purified hepatic cytochrome P-450 from uninduced mice
Different effects of local anesthetics on calcium influx into rat mast cells
Isoproterenol-sensitive adenylate cyclase in glomeruli iso- lated from young and adult rat renal cortex
Studies of [3H]nitrendipine binding and KCl-induced calcium uptake in rat cortical synaptosomes
Effects of calcium antagonists on smooth muscle membranes of the canine stomach
Aluminum intake from non-prescription drugs and sucralfate
Disparate responses of blood pressure to adrenergic stimuli during beta blockade
Effect of adenosine 5'-triphosphate (ATP) on the isolated rectum of the rainbow lizard Agama agama
Evidence for multiple sources of calcium involved on the contractile effects of agonists in the dog uterus. Influence of ovarian sexual hormones
Effect of tetraethylammonium and verapamil on nor- adrenaline release induced by field electrical stimulation and potassium from cat cerebral and femoral arteries
Dose-related effects of fentanyl on autonomic and behavioral responses in performance horses
Study of fl-adrenoceptors and fl-adrenergic responsiveness in cultured "'preneoplastic-like" and neoplastic rat hepatocytes
A beta-adrenoceptor blocking agent, befunolol as a partial agonist in isolated organs
269 Interaction of muscarinic drugs with their receptor
Yoshiaki Akimoto, Hitoshi Nishimura, Masamichi Komiya, Tomomi Shibata, Kenji Kaneko, Akira Fujii and Toyoyuki Tamura
V. Bocci, G. P. Pessina, A. Pacini, L. Paulesu, M. Muscettola, A. Naldini and G. Lunghetti
Takeshi Katsuragi, Kazuo Furuta, Toshiro Harada and Tatsuo Furukawa
273
277
281
Concentrations of ampicillin and cefadroxil in human serum and mixed saliva following a single oral administration of talampicillin and cefadroxil, and relationships between serum and mixed saliva concentrations
Pharmacokinetics of human lymphoblastoid interferon in rabbits
A possible explanation for a greater discrepant suppression by adenosine and N6-cyclohexyl adenosine of the guinea-pig ileal contraction
S. Evangelista and A. Meli
Jos~ Ram6n Naranjo, Mario Fernandez-Roman, Maria del Carmen Urdin and Jos~ A. Fuentes
Gary B. Giavin
Ewa Turska, Lilla Lachowicz, Wiktor Kozioikiewicz and Tadeusz Wasiak
S. Gottfried~.I~, R. S. Vine and B. Y. C. Wan
B. M. Faggin and J. Palermo-Neto
M. Ubeda, F. Fenoy, L. F. Carbonell, F. J. Salazar, J. Garcia-Estafi, M. G. Salom and T. Quesada
285
287
Influence of antioxidants and radical scavengers on ethanol- induced gastric ulcers in the rat
/~-endorphin: a common factor in the antihypertensive action of clonidine-type imidazolines in spontaneously hypertensive rats
291 Zinc sulphate reduces activity-stress gastric lesions in rats
293 Effects of analogues of substance P fragments on the MAO activity in rat brain
297
299
A quantitative morphological study of the effects of car- benoxolone sodium on duodenal goblet-cells of the rat
Differential alterations in brain sensitivity to amphetamine and pentylenetetrazol in socially deprived mice
303 Effect of captopril on norepinephrine vascular contractility
Minireview
James R. Jauchem 307
Vol. 16, No. 4
Effects of drugs on thermal responses to microwaves
General Papers
P. V. Sulakhe, N. T. Phan and G. Jagadeesh
Terry L. Johnson and Charles O. Knowles
Koki Kato and Hideomi Fukuda
Kazuhiko Ohishi, Tamiko Suzuki and Masaatsu K. Uchida
Sumantra Das and Hemendra N. Bhargava
Thomas Yorio, Ron Royce, Janet Mattern, Larry X. Oakford, A. J. Mia and Nimman Tarapoom
M. F. Kenel and A. P. Kulkarni
311 Comparison of cholinergic inihibition and beta-adrenergic stimulation of adenylate cyclase from rat and guinea-pig hearts: effects of guanine nucleotides and monovalent cations
321 Formamidine-mediated inhibition of rat platelet aggregation
327
335
341
347
355
The non-GABAergic nature of 3H-baclofen binding in rat peripheral tissues
Relation between inhibition of calmodulin and mediator release from rat mast cells
Effect of prolyl-leucyl-glycinamide on blood pressure, heart rate and angiotensin converting enzyme activity in spontane- ously hypertensive and Wistar-Kyoto normotensive rats
Inhibition of the hydro-osmotic response to vasopressin and hypertonicity by phenothiazines and W7, calmodulin antagonists
Ethanol potentiation of carbon tetrachloride hepatotoxicity: possible role for the in vivo inhibition of aldehyde dehydrogenase
Markku Pasanen and Olavi Pelkonen 361 Resolution of multiple P-450 forms: separation of aryl hydrocarbon hydroxylase and aminopyrine N-demethylase- associated P-450 isoenzymes by chromatofocusing
D. R. Mottram and P. Saggar 367 Cirazoline, an :~2-adrenoceptor antagonist in guinea-pig ileum
M. H. Hawthorn, K. J. Broadley and C. J. Gibbon
371 Examination of the bronchoconstrictor response of guinea- pig isolated lung to /3-phenylethylamine
Fukio Konno, Yuka Sato, Kunimi Togashi, lssei Takayanagi and Masaaki Hirobe
379 Interactions of codeine-7,8-oxide (codeine-epoxide), as a new metabolite of codeine, with multiple opiate receptors
Minoru Tanaka and Yasuko Shibata 383 The different response of guinea pig peritoneal macrophages to various stimulators
C. Nze. Aguwa 387 Gastrointestinal effects of the extracts of Rhigiocarya racem- (fera ( Menispermaceae )
Nobuhiro Satake, Shoichi Ueda and Shoji Shibata
391 Dopamine-induced potentiation of the contractile response to arachidonic acid in guinea-pig aorta
N. D. Vaziri and C. Byrne 395 Effects of glucose feeding on renal electrolyte and H ~ transport
Jos~ Carlos Gomes and Abilio Antonio 399 Histamine release from the isolated guinea-pig heart by compound 48/80
Maria M. Bernardi, Moacyr L. Aizenstein, Roberto DeLucia and Crist6foro Scavone
403 Influence of phenoxybenzamine on the stereotyped behaviour induced by fencamfamine in rats: evidence for a qualitative alteration
Maria M. Bernardi and Crist6foro Scavone
407 Differential biochemical and behavioral effects of single and chronic administration of amphetamine and apomorphine
P. Garz6n, S. Gonzfilez-Cornejo, S. Romfin-Maldonado and A. Navarro-Ruiz
411 Valproic acid and phenytoin effects on serum proteins and immunoglobulins of epileptic patients
Francesc Villarroya and Teresa Mampel
415 Glucose tolerance and insulin response in offspring of ethanol-treated pregnant rats
Antonio Chapola, Nelson Villa, Luiz B. S. Valle, Ricardo M. Oliveira-Filho and Conceiq~o A. S. A. Minetti
419 fl-adrenergic stimulation of mouse parotid gland: amylase activity and secretory granules during isoproterenol-induced mitosis
C. Almodovar-Cuevas, A. Navarro-Ruiz, B. E. Bastidas-Ramirez, Ma. R. Mora-Navarro and P. Garz6n
423 Valproic acid effects on leukocytes and platelets of Sprague-Dawley rats
Book Reviews 427
New Patents i New patents and published patent applications from the United States and over 30 other countries
Review
G. Burnstock and C. Kennedy
Minireview
Edward J. Hammond and B. J. Wilder
Vol. 16, No. 5
433 Is there a basis for distinguishing two types of P2-purino- ceptor?
441 Gamma-vinyl GABA
vii
General Papers Masaatsn-Koujirou Uchida and Mitsuo Mita
Shunzo Nishibe, Michio Ogawa, Goro Kosaki and Takesada Mori
Antonio R. Granata
C. F. Sfinchez-Ferrer, J. Marin, M. Salaices, M. L. Rico and J. L. Mufioz-Blanco
Lynn Bradley and Sheila A. Doggrell
T. R. Hall, S. Harvey and A. Chadwick
Carlos Beas-Zfirate, Jorge Arauz-Contreras, Anselmo Velazquez and Alfredo Feria-Velasco
M. J. Carmena and J. C. Prieto
I. Takayanagi, F. Konno and M. Kusunoki
J. S. Serrano, F. J. Mifiano, M. Saneibrifin and J. A. Durfin
N. Seiler, S. Sarhan, P. Krogsgaard-Larsen, H. Hjeds and A. Schousboe
Tetsnyuki Nasu, Kazuyoshi Gyobn and Yukio Ishida
S. C. Yeong and A. V. Jnorio
Robin A. Barraco, John W. Phillis and Harvey J. Altman
Charles D. Lox, Dennis M. Lox and M. Wayne Heine
E. Contreras and L. Tamayo
H. De Souza and J. Palermo-Neto
Francesc Villarroya, Teresa Mampel and Emilio Herrera
449
455
463
469
475
483
489
495
501
505
509
513
517
521
Effects of Quin-2, an intracellular Ca chelator, and TMB-8, an intracellular Ca antagonist, on the short-term desensi- tization to histamine in guinea pig taenia caecum
Effects of protease inhibitors and calmodulin inhibitors on Ca 2+ influx and catecholamine secretion in isolated bovine adrenal medullary cells
Prolonged treatment with (_+)propranolol induces super- sensitivity to (L)noradrenaline in mesenteric arteries in the rat
Interference of pentobarbital and thiopental with the vascu- lar contraction and noradrenaline release in human cerebral arteries
Modification of desipramine of the effects of ~-adrenoceptor antagonists on the contractile responses of the trisected rat vas deferens
Effects of putative neurotransmitters on release of prolactin from pituitary glands of the domestic fowl co-incubated with hypothalamic tissue
Monosodium L-glutamate-induced convulsions II. Changes in catecholamine concentrations in various brain areas of adult rats
VIP binding to epithelial cell membranes of rat ventral prostate: effect of guanine nucleotides
Some pharmacological effects of tizanidine on smooth muscle organs and ~:-adrenoceptor
Involvement of bicuculline-insensitive receptors in the hypo- thermic effect of GABA and its agonists
Amplification by glycine of the anticonvulsant effect of THPO, a GABA uptake inhibitor
Analysis of mercury ions binding to the smooth muscle of guinea-pig taenia coli
The effects of estradiol and progesterone on the concen- tration of striatal dopamine and tyramine in ovariectomized mice
Depressant effect of forskolin on spontaneous locomotor activity in mice
525 Effects of acute ethanol intoxication combined with seco- barbital abuse on hemostasis
529 Effects of ethylenediamine on morphine analgesia and tolerance-dependence in mice
533 A biochemical study of cholinergic dopaminergic inter- actions in the central nervous system
537 Similar metabolic response to acute ethanol intake in preg- nant and non-pregnant rats either fed or fasted
viii
Ghandi M. Saadeh, Raja E. Ayash, Fadi M. Saadeh and Camille F. Nassar
Book Reviews
541
545
Effect of aminophylline on calcium transport across the rat diaphragm
Minireviews T. B. Ng and H. W. Yeung
F. V. DeFeudis
General Papers
M. S. Dar, P. L. Morselli and E. R. Bowman
Gabriella Coruzzi, Enzo Poli and Giulio Bertaccini
Maria E. M. Oshiro, Antonio C. M. Paiva and Therezinha B. Paiva
Helen Kotsifaki, Vasilios Kapoulas and George Deliconstantinos
Carlo Alberto Maggi, Sandro Giuliani and Alberto Meli
Lorie R. Pelc, Garrett J. Gross and David C. Warltier
Francesc Villarroya and Teresa Mampel
I. N. Stoyanov, K. T. Milenov, A. G. Ter-Margaryan, M. P. Milanov and V. I. Vassilev
R. C. Elliott
J. W. Phillis, A. S. Bender and W. Marszalec
I. Takayanagi, F. Konno, H. Arai, K. Chimoto and T. Kitada
I. Takayanagi, K. Okumura, F. Konno, K. Koike, N. Cho and M. Hirobe
P. S. Key, N. D. Vaziri and M. Childester
Camille F. Nassar, Michel G. Nasser and Zouheir M. Habbal
Vol. 16, No. 6
549 Hypoglycemic constituents of Panax ginseng
553 Are vascular mechanisms involved in antidepressant action?
557
561
567
573
579
The enzymatic systems involved in the mammalian metabo- lism of methylamine
Action of different agonists and antagonists of the cholinergic system on the rat lower esophageal sphincter
Endothelium-dependent inhibition of the use of extracellular calcium for the arterial response to vasoconstrictor agents
Targeting of liposomes containing methotrexate towards Tetrahymena pyriformis cells
The effect of peripherally administered GABA on noradren- aline-induced reflex vagal bradycardia in urethane ana- esthetized rats
585 Cardiac and systemic hemodynamic actions of the slow channel calcium blocking agent, KB-944
591
597
603
609
613
617
621
625
Effects of chronic ethanol treatment on glucose tolerance, insulin response and circulating metabolites in the pregnant rat
Effects of prostaglandin F2~ and indomethacin on the contractile activity of different compartments of the complex stomach
The action of intravenous anaesthetic and central depressant drugs on the contractures elicited by tetraethylammonium in the chick biventer cervicis muscle
Estradiol and progesterone potentiate adenosine's depressant action on rat cerebral cortical neurons
Newly synthesized ~l-adrenoceptor blockers (SM911 and SM2470) and characterization of ct-adrenoceptors in rat aortic strips, rat vas deferens preparations and rabbit aortic strips
Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13,nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor
Effect of H 2 histamine receptor blockade and stimulation on urinary acidification
Receptors of prostaglandin E l in the plasma membrane of normal liver. Effect of membrane fluidity on PGE~ binding
ix
C. P~rez, M. E. Otero Losada and 629 M. C. Rubio
M. Salaices, A. de Gregorio 633 and J. Matin
Seico Hanada, Seizi Oga and Marcia T. Hirano
B. Bouscarel, J. C. Murat and H. Paris 641
Book Reviews 645
Changes in GABAergic system parameters after chronic administration of bicuculline
Study of vasodilator effects of papaverine, adenosine and related drugs in isolated cat cerebral arteries
637 Some characteristics of econazole-induced pleurisy in rats
Involvement of guanine nucleotide and sodium in regulation of yohimbine and clonidine binding sites in the HT29 human colon adenocarcinoma cell-line