ChemInform Abstract: Palladium-Catalyzed Direct Oxidative Heck—Cassar—Sonogashira Type...

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ChemInform 2010, 41, issue 44 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim www.cheminform.wiley-vch.de Indole derivatives R 0140 DOI: 10.1002/chin.201044111 Palladium-Catalyzed Direct Oxidative Heck—Cassar—Sonogashira Type Alky- nylation of Indoles with Alkynes under Oxygen. — Unlike previous methods, the ti- tle reaction does not need the pregeneration of indolyl or alkynyl halide. Furthermore, only a catalytic amount of base is required and oxygen is used as the terminal oxidant. — (YANG, L.; ZHAO, L.; LI*, C.-J.; Chem. Commun. (Cambridge) 46 (2010) 23, 4184-4186, DOI:10.1039/c0cc00014k ; Dep. Chem., McGill Univ., Montreal, Que. H3A 2K6, Can.; Eng.) — M. Paetzel 44- 111

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Indole derivativesR 0140 DOI: 10.1002/chin.201044111

Palladium-Catalyzed Direct Oxidative Heck—Cassar—Sonogashira Type Alky-nylation of Indoles with Alkynes under Oxygen. — Unlike previous methods, the ti-tle reaction does not need the pregeneration of indolyl or alkynyl halide. Furthermore, only a catalytic amount of base is required and oxygen is used as the terminal oxidant. — (YANG, L.; ZHAO, L.; LI*, C.-J.; Chem. Commun. (Cambridge) 46 (2010) 23, 4184-4186, DOI:10.1039/c0cc00014k ; Dep. Chem., McGill Univ., Montreal, Que. H3A 2K6, Can.; Eng.) — M. Paetzel

44- 111

ChemInform 2010, 41, issue 44 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

ChemInform RxnFinder

ChemInform RxnFinder

RESEARCHARTICLE LargescalecomparisonofQSAR … · 2020. 3. 19. · Boscet al. J Cheminform Page3of16 Dta preparation Compoundstructureswereextractedfromthedatabase inSMILESformatandusingRDKit(version2017_09_01)

RESEARCHARTICLE LargescalecomparisonofQSAR … · 2020. 3. 19. · Boscet al. J Cheminform Page3of16 Dta preparation Compoundstructureswereextractedfromthedatabase inSMILESformatandusingRDKit(version2017_09_01)

GPURFSCREEN: a GPU based virtual screening tool …people.cse.nitc.ac.in/jayaraj/files/gpurfscreen...Jayaraj et al. J Cheminform DOI 10.1186/s13321-016-0124-8 SOFTWARE GPURFSCREEN:

GPURFSCREEN: a GPU based virtual screening tool …people.cse.nitc.ac.in/jayaraj/files/gpurfscreen...Jayaraj et al. J Cheminform DOI 10.1186/s13321-016-0124-8 SOFTWARE GPURFSCREEN:

OSYNTHESIS-Heck - Sonogashira - Stille - Suziki Cross Coupling Reactions

OSYNTHESIS-Heck - Sonogashira - Stille - Suziki Cross Coupling Reactions

MER: a shell script and annotation server for minimal named ......Couto and Lamurias J Cheminform Page 5 of 10 common,sandswesempiricallysfoundsthatsmostsofsthestwo-charactersmatchesswereserrors

MER: a shell script and annotation server for minimal named ......Couto and Lamurias J Cheminform Page 5 of 10 common,sandswesempiricallysfoundsthatsmostsofsthestwo-charactersmatchesswereserrors

PART I€¦ · Stille, Heck, Suzuki, Sonogashira, Kumada, Negishi, Nozaki–Hiyama, Buchwald–Hartwig, and Tsuji–Trost [13]. These reactions are usually very efficient, although

PART I€¦ · Stille, Heck, Suzuki, Sonogashira, Kumada, Negishi, Nozaki–Hiyama, Buchwald–Hartwig, and Tsuji–Trost [13]. These reactions are usually very efficient, although

Synthesis of Carbohydrate Fused Chiral Macrocyclic ... Synthesis of Carbohydrate Fused Chiral Macrocyclic Benzolactones through Sonogashira Reaction Altaf Hussain, 1,2 1,2Mallikharjuna

Synthesis of Carbohydrate Fused Chiral Macrocyclic ... Synthesis of Carbohydrate Fused Chiral Macrocyclic Benzolactones through Sonogashira Reaction Altaf Hussain, 1,2 1,2Mallikharjuna

Stille, Suzuki, and Sonogashira Couplings Cross-Coupling ...tminehan.com/531pdfs2/StilleSuzuki.pdf · Suzuki Coupling Suzuki Coupling is the reaction of vinyl or aryl boronic acids

Stille, Suzuki, and Sonogashira Couplings Cross-Coupling ...tminehan.com/531pdfs2/StilleSuzuki.pdf · Suzuki Coupling Suzuki Coupling is the reaction of vinyl or aryl boronic acids

Carbonylative Sonogashira coupling of Benzyl chlorides … · Supporting Information Palladium-Catalyzed Carbonylative Coupling of Benzyl Chlorides with Terminal Alkynes to 1,4-Diaryl-3-butyn-2-ones

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METHODOLOGY Ecientiterativevirtualscreening with … · 2018. 3. 1. · Ahmed et al. J Cheminform Page4of8 10contain‘high-scoring’ligands.eunassignedbin3is excludedfromtraining.Figure

METHODOLOGY Ecientiterativevirtualscreening with … · 2018. 3. 1. · Ahmed et al. J Cheminform Page4of8 10contain‘high-scoring’ligands.eunassignedbin3is excludedfromtraining.Figure

Method Development, Synthesis and Mechanistic · 2013. 10. 3. · cycloparaphenylenes via Sonogashira cross-coupling reactions and [2+2+2]-cycloadditions. After some preliminary experiments

Method Development, Synthesis and Mechanistic · 2013. 10. 3. · cycloparaphenylenes via Sonogashira cross-coupling reactions and [2+2+2]-cycloadditions. After some preliminary experiments

Alkynylation of Terminal Alkynes with Alkynyl Hypervalent ...acetylene gold intermediate 14 to the silver(I)-activated alkynyl hypervalent iodine (6) along pathway IV shown in Scheme

Alkynylation of Terminal Alkynes with Alkynyl Hypervalent ...acetylene gold intermediate 14 to the silver(I)-activated alkynyl hypervalent iodine (6) along pathway IV shown in Scheme

Database fingerprint (DFP): an approach to represent ... · Fernández‑de Gortari et al. J Cheminform DOI 10.1186/s13321‑017‑0195‑1 PRELIMINARY COMMUNICATION Database fingerprint

Database fingerprint (DFP): an approach to represent ... · Fernández‑de Gortari et al. J Cheminform DOI 10.1186/s13321‑017‑0195‑1 PRELIMINARY COMMUNICATION Database fingerprint

Sonogashira Mechanisms

Sonogashira Mechanisms

c Consult author(s) regarding copyright matterseprints.qut.edu.au › 30665 › 1 › The_Palladium-Catalysed... · The Palladium-Catalysed Copper-Free Sonogashira Coupling of Isoindoline

c Consult author(s) regarding copyright matterseprints.qut.edu.au › 30665 › 1 › The_Palladium-Catalysed... · The Palladium-Catalysed Copper-Free Sonogashira Coupling of Isoindoline

Direct Alkynylation of Thiophenes: Cooperative Activation ...propylsilyl)buta 1,3 diyne, and no strong effect of TFA was observed. [23] No Au-bond intermediate could be detected. These

Direct Alkynylation of Thiophenes: Cooperative Activation ...propylsilyl)buta 1,3 diyne, and no strong effect of TFA was observed. [23] No Au-bond intermediate could be detected. These

Supporting information prepared by Sonogashira dispersion polymerization … · 2015. 5. 1. · while the tip sonicator was running consistently at 12 W. all the catalyst had dissolved,

Supporting information prepared by Sonogashira dispersion polymerization … · 2015. 5. 1. · while the tip sonicator was running consistently at 12 W. all the catalyst had dissolved,

Investigation of Low-Dimensional Conjugated Nanostructures on … · 2019. 9. 6. · Sonogashira cross-coupling Au(100) On-surface SCC coupling only took place at island boundaries.

Investigation of Low-Dimensional Conjugated Nanostructures on … · 2019. 9. 6. · Sonogashira cross-coupling Au(100) On-surface SCC coupling only took place at island boundaries.

Ligand-, Copper-, and Amine-Free Sonogashira Reaction of Aryl

Ligand-, Copper-, and Amine-Free Sonogashira Reaction of Aryl

BROMOTRYPTOPHANS AND THEIR INCORPORATION IN …diposit.ub.edu/dspace/bitstream/2445/121062/1/679729.pdfor Pd-catalyzed Sonogashira reactions. Owing to the great interest in tryptophan

BROMOTRYPTOPHANS AND THEIR INCORPORATION IN …diposit.ub.edu/dspace/bitstream/2445/121062/1/679729.pdfor Pd-catalyzed Sonogashira reactions. Owing to the great interest in tryptophan