ChemInform Abstract: An Expeditious Synthesis and Anticancer Activity of Novel...

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ChemInform 2010, 41, issue 28 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim www.cheminform.wiley-vch.de Oxazole derivatives R 0220 DOI: 10.1002/chin.201028127 An Expeditious Synthesis and Anticancer Activity of Novel 4-(3'-Indolyl)oxazoles. — Novel indolyloxazoles such as (VI) and (VIII) are synthesized via microwave- -accelerated reaction of tosyloxyacetylindole (III) with amides. Compounds (VIh) and (VIII) are found to be most cytotoxic and selective against various cancer cell lines. — (KUMAR*, D.; KUMAR, N. M.; SUNDAREE, S.; JOHNSON, E. O.; SHAH, K.; Eur. J. Med. Chem. 45 (2010) 3, 1244-1249; Chem. Group, Birla Inst. Technol. Sci., Pilani 333 031, India; Eng.) — H. Toeppel 28- 127

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Oxazole derivativesR 0220 DOI: 10.1002/chin.201028127

An Expeditious Synthesis and Anticancer Activity of Novel 4-(3'-Indolyl)oxazoles. — Novel indolyloxazoles such as (VI) and (VIII) are synthesized via microwave--accelerated reaction of tosyloxyacetylindole (III) with amides. Compounds (VIh) and (VIII) are found to be most cytotoxic and selective against various cancer cell lines. — (KUMAR*, D.; KUMAR, N. M.; SUNDAREE, S.; JOHNSON, E. O.; SHAH, K.; Eur. J. Med. Chem. 45 (2010) 3, 1244-1249; Chem. Group, Birla Inst. Technol. Sci., Pilani 333 031, India; Eng.) — H. Toeppel

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ChemInform 2010, 41, issue 28 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

TRANSITION METAL-MEDIATED SYNTHESIS OF OXAZOLES … · oxazole ring. The majority of these transformations, driven by the transition metal complexes, involve nucleophilic additions

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IDENTIFICATION OF OUTLIERS IN OXAZOLINES AND OXAZOLES HIGH DIMENSION MOLECULAR DESCRIPTOR DATASET USING PRINCIPAL COMPONENT OUTLIER DETECTION ALGORITHM AND COMPARATIVE NUMERICAL STUDY

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STUDY OF NOVEL SYNTHETIC METHODOLOGIES FOR INDOLYL ...

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NMDA receptor antagonism with novel indolyl, 2-(1,1 ...

Classification System for Solid Supports Used ... - FIZ CHEMIE › fileadmin › user_upload › Cheminform › Spore › _… · FIZ CHEMIE BERLIN - 5 (23) - The remainder of the

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Oxidation of 4-(3-Indolyl)- and 4-(5-Indolyl)-1,4 ...

ChemInform Sheet A4 · 2013. 9. 13. · The ChemInform Reaction Library (CIRX) helps to deal with the enormous number of published reactions as it does not cover all information available

ChemInform Sheet A4 · 2013. 9. 13. · The ChemInform Reaction Library (CIRX) helps to deal with the enormous number of published reactions as it does not cover all information available

Continuous multistep synthesis of 2-(azidomethyl)oxazoles€¦ · 506 Continuous multistep synthesis of 2-(azidomethyl)oxazoles Thaís€A.€Rossa1,2, Nícolas€S.€Suveges3, Marcus€M.€Sá2,

Continuous multistep synthesis of 2-(azidomethyl)oxazoles€¦ · 506 Continuous multistep synthesis of 2-(azidomethyl)oxazoles Thaís€A.€Rossa1,2, Nícolas€S.€Suveges3, Marcus€M.€Sá2,

Fine Chemicals · 2019. 11. 28. · Indoles, Benzindoles 17 Imidazoles, Pyrazoles 18. Triazoles 19. Tetrazoles 20. Oxazoles 21. Selenazoles, Thiazoles 22. Piperidines, Pyridines,

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Performance analysis of neural network models for oxazolines and oxazoles derivatives descriptor dataset

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BIOINFORMATICS Review …“.Jónsdóttir et al. Fig. 1. Number of papers in PubMed 1992–2004 containing the keywords ‘bioinformatics’ (top left), ‘chemoinformatics’ or ‘cheminform-atics’,

BIOINFORMATICS Review …“.Jónsdóttir et al. Fig. 1. Number of papers in PubMed 1992–2004 containing the keywords ‘bioinformatics’ (top left), ‘chemoinformatics’ or ‘cheminform-atics’,

RESEARCHARTICLE OpAccess ......Jiangiet al. J Cheminform Pagej2jofj26 playerindrugabsorption,distribution,metabolism, excretion,andtoxicity(ADMET)[5, 6],andhasalsobeen ...

RESEARCHARTICLE OpAccess ......Jiangiet al. J Cheminform Pagej2jofj26 playerindrugabsorption,distribution,metabolism, excretion,andtoxicity(ADMET)[5, 6],andhasalsobeen ...

Heterocyclic Compoundsmu-varna.bg/EN/Students/Documents/organic-chemistry/... · Web viewOther indolic compounds include the plant hormone Auxin (indolyl-3-acetic acid, IAA), the

Heterocyclic Compoundsmu-varna.bg/EN/Students/Documents/organic-chemistry/... · Web viewOther indolic compounds include the plant hormone Auxin (indolyl-3-acetic acid, IAA), the

ChemInform Sheet A4on chemo-, regio-, and stereo-selective reactions. The RefLib database is included with CIRX and provides reactions abstracted from Theilheimer’s Synthetic Methods

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Compounds related to 3-alkylamine-1H-indolyl acrylate and ...

 · Esterilidad Comercial Aerobios mesófilos (Conteo en placa) Clostridium peffnnges ... technique at 44 0 C using 5-bromo -4 chloro-3 indolyl -B-D-glucoronide.

 · Esterilidad Comercial Aerobios mesófilos (Conteo en placa) Clostridium peffnnges ... technique at 44 0 C using 5-bromo -4 chloro-3 indolyl -B-D-glucoronide.