A Formal [3 + 2] Cycloaddition Process with Nonactivated Aziridines to Polysubstituted...

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2006 Fused pyridine derivatives R 0450 A Formal [3 + 2] Cycloaddition Process with Nonactivated Aziridines to Polysub- stituted Indolizidines. — A sequential SN2/[3 + 2] cycloaddition process affords a va- riety of indolizidines in moderate to good yields. The chiral version of the reaction is demonstrated to proceed with complete chirality transfer. — (ZHU, W.; CAI, G.; MA*, D.; Org. Lett. 7 (2005) 25, 5545-5548; State Key Lab. Bioorg. Nat. Prod. Chem., Shanghai Inst. Org. Chem., Acad. Sin., Shanghai 200032, Peop. Rep. China; Eng.) — R. Steudel 17- 155

Transcript of A Formal [3 + 2] Cycloaddition Process with Nonactivated Aziridines to Polysubstituted...

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2006

Fused pyridine derivativesR 0450 A Formal [3 + 2] Cycloaddition Process with Nonactivated Aziridines to Polysub-

stituted Indolizidines. — A sequential SN2/[3 + 2] cycloaddition process affords a va-riety of indolizidines in moderate to good yields. The chiral version of the reaction is demonstrated to proceed with complete chirality transfer. — (ZHU, W.; CAI, G.; MA*, D.; Org. Lett. 7 (2005) 25, 5545-5548; State Key Lab. Bioorg. Nat. Prod. Chem., Shanghai Inst. Org. Chem., Acad. Sin., Shanghai 200032, Peop. Rep. China; Eng.) — R. Steudel

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O Syntheses of Aziridines OY O O R Me N NH Z Me N N Me N ...gbdong.cm.utexas.edu/seminar/old/Syntheses of Aziridines_Haye Mi… · Syntheses of Aziridines 2014. 03. 05 Haye Min Ko

O Syntheses of Aziridines OY O O R Me N NH Z Me N N Me N ...gbdong.cm.utexas.edu/seminar/old/Syntheses of Aziridines_Haye Mi… · Syntheses of Aziridines 2014. 03. 05 Haye Min Ko

Stereoselective Routes to Aziridines Nate Bowling McMahon Group University of Wisconsin-Madison Sept. 12, 2002.

Stereoselective Routes to Aziridines Nate Bowling McMahon Group University of Wisconsin-Madison Sept. 12, 2002.

Microwave-assisted regioselective ring opening of non-activated aziridines by lithium ... · Microwave-assisted regioselective ring opening of non-activated aziridines by lithium

Microwave-assisted regioselective ring opening of non-activated aziridines by lithium ... · Microwave-assisted regioselective ring opening of non-activated aziridines by lithium

Straightforward synthesis of 1-alkyl-2-(trifluoromethyl ...An efficient and straightforward approach towards the synthesis of 1-alkyl-2-(trifluoromethyl)-aziridines starting from 1,1,1-trifluoroacetone

Straightforward synthesis of 1-alkyl-2-(trifluoromethyl ...An efficient and straightforward approach towards the synthesis of 1-alkyl-2-(trifluoromethyl)-aziridines starting from 1,1,1-trifluoroacetone

The role of polysubstituted heterocycles in the synthesis ... N-Heteroarylformamidines, N-heteroarylacetamidines, N-heteroarylform-amide oximes, and N-heteroarylacetamide oximes are

The role of polysubstituted heterocycles in the synthesis ... N-Heteroarylformamidines, N-heteroarylacetamidines, N-heteroarylform-amide oximes, and N-heteroarylacetamide oximes are

Northumbria Research Linknrl.northumbria.ac.uk/38425/1/Chem_Eur_J_2016_author_accepted.pdfReactions in Photochemically-Generated Vinyl Aziridines Jonathan P. Knowles*[a] and Kevin

Northumbria Research Linknrl.northumbria.ac.uk/38425/1/Chem_Eur_J_2016_author_accepted.pdfReactions in Photochemically-Generated Vinyl Aziridines Jonathan P. Knowles*[a] and Kevin

One-pot Multi-component Synthesis of Some ... · PDF filesynthesis of polysubstituted imidazoles via one-pot multi-component reaction of various aldehydes, benzil, aliphatic/aromatic

One-pot Multi-component Synthesis of Some ... · PDF filesynthesis of polysubstituted imidazoles via one-pot multi-component reaction of various aldehydes, benzil, aliphatic/aromatic

Ring Expansions of Vinyloxiranes, -thiiranes, and -aziridines: …szolcsanyi/education/files/Chemia... · 2013. 10. 28. · to many useful synthetic intermediates. This paper highlights

Ring Expansions of Vinyloxiranes, -thiiranes, and -aziridines: …szolcsanyi/education/files/Chemia... · 2013. 10. 28. · to many useful synthetic intermediates. This paper highlights

One-pot Synthesis of Polysubstituted Dihydro-2- oxypyrroles …jacr.kiau.ac.ir/article_527186_4f621a6e88516fd2b8485bca4... · 2020-06-23 · low-cost, eco-friendly, one-pot, simple

One-pot Synthesis of Polysubstituted Dihydro-2- oxypyrroles …jacr.kiau.ac.ir/article_527186_4f621a6e88516fd2b8485bca4... · 2020-06-23 · low-cost, eco-friendly, one-pot, simple

Asymmetric synthesis of CF2-functionalized aziridines by combined strong Brønsted ... · 2020-04-07 · 638 Asymmetric synthesis of CF2-functionalized aziridines by combined strong

Asymmetric synthesis of CF2-functionalized aziridines by combined strong Brønsted ... · 2020-04-07 · 638 Asymmetric synthesis of CF2-functionalized aziridines by combined strong

Cycloaddition [3+2] de cétènes avec des aziridines

Cycloaddition [3+2] de cétènes avec des aziridines

Evolution of metastases-associated fibroblasts in the lung ... · secreted factors significantly enhanced the capacity of to contract collagen gels as NLF compared with control nonactivated

Evolution of metastases-associated fibroblasts in the lung ... · secreted factors significantly enhanced the capacity of to contract collagen gels as NLF compared with control nonactivated

Employing Carboxylic Acids in Aryne Multicomponent ... · Employing Carboxylic Acids in Aryne Multicomponent Coupling Triggered by Aziridines/Azetidines ... distillation over Na-benzophenone

Employing Carboxylic Acids in Aryne Multicomponent ... · Employing Carboxylic Acids in Aryne Multicomponent Coupling Triggered by Aziridines/Azetidines ... distillation over Na-benzophenone

Table of Contents1 . Cascade reactions of indi go with oxiranes and aziridines: efficient access to dihydropyrazinodiindoles and spiro -oxazocinodiindoles. Nicholas M. Butler, Rudi

Table of Contents1 . Cascade reactions of indi go with oxiranes and aziridines: efficient access to dihydropyrazinodiindoles and spiro -oxazocinodiindoles. Nicholas M. Butler, Rudi

Protein Components of the Nonactivated Glucocorticoid Receptor* · 2001-06-12 · p59-specific signal with the molybdate-stabilized receptor and only a very faint band in the material

Protein Components of the Nonactivated Glucocorticoid Receptor* · 2001-06-12 · p59-specific signal with the molybdate-stabilized receptor and only a very faint band in the material

RadicalCationsofPhenyl-Substituted Aziridines: What are ...

RadicalCationsofPhenyl-Substituted Aziridines: What are ...

AgOTf-Catalyzed dehydrative [3+2] annulation of aziridines ... · S1 AgOTf-Catalyzed dehydrative [3+2] annulation of aziridines with 2-naphthols Trinadh Kaicharla,a,b Anu Jacob,a

AgOTf-Catalyzed dehydrative [3+2] annulation of aziridines ... · S1 AgOTf-Catalyzed dehydrative [3+2] annulation of aziridines with 2-naphthols Trinadh Kaicharla,a,b Anu Jacob,a

Synthesis and Safety - John Wiley & Sonscatalogimages.wiley.com/images/db/pdf/9780470519981.excerpt.pdf · nitrenium ions as well as nitrogen - rich compounds such as aziridines,

Synthesis and Safety - John Wiley & Sonscatalogimages.wiley.com/images/db/pdf/9780470519981.excerpt.pdf · nitrenium ions as well as nitrogen - rich compounds such as aziridines,

Catalytic Asymmetric Synthesis of Trisubstituted Aziridines

Catalytic Asymmetric Synthesis of Trisubstituted Aziridines

The role of polysubstituted heterocycles in the synthesis ... phosphorous trichloride. With acetic anhydride they can be rearranged into the corresponding 2-acetoxy derivatives 10

The role of polysubstituted heterocycles in the synthesis ... phosphorous trichloride. With acetic anhydride they can be rearranged into the corresponding 2-acetoxy derivatives 10