2003-2004 Review of Anticoagulants, Thrombolytics and Anti-platelet Drugs 3 November 2015 5:19 AM.
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Transcript of 2003-2004 Review of Anticoagulants, Thrombolytics and Anti-platelet Drugs 3 November 2015 5:19 AM.
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2003-2004Review of Anticoagulants,
Thrombolytics and Anti-platelet Drugs
April 20, 202306:30 AM
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Abciximab
Antiplatelet
Anti-GPIIb/IIIa receptor antibody
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Adalimumab
TNF inhibitor
Anti-TNF antibodyUsed in rheumatoid arthritis
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Allopurinol
AntigoutAntineoplastic (supporting
agent)
Folic acid analogueXanthine oxidase inhibitor
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Aminocaproic acid (EACA)
Procoagulant
Inhibitor of plasminogen activation
(decreases fibrinolysis)
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Anistreplase
Thrombolytic
Streptokinase + plasminogen
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Aprotinin
Procoagulant
Fibrinolytic inhibitorSerine protease inhibitor
(“serpin”)Streptokinase inhibitor
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Argatroban
Anticoagulant
Direct thrombin inhibitor
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Aspirin(Acetylsalicylic acid, ASA)
NSAID (acetylsalicylate)Analgesic, Anti-inflammatory
Antipyretic, Antiplatelet
Irreversible cyclooxygenase inhibitor
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Atorvastatin
Antihyperlipidemic
HMG-CoA reductase inhibitor
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Auranofin
Disease modifyinganti-rheumatic drug (DMARD)
Gold saltOral
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Aurothioglucose
Disease modifyinganti-rheumatic drug (DMARD)
Gold saltParenteral
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Balsalazide
NSAID (salicylate)
Treatment of IBD
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Beclomethasone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled
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Betamethasone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidNot by inhalation
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Bivalirudin
Anticoagulant
Direct thrombin inhibitor
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Bradykinin
Inflammatory mediator
Plasma, hypotension, pain
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Budesonide
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled OR treatment of IBD
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C3a, C5a
Inflammatory mediators
Anaphylatoxins Low molecular weight
complement cleavage products
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Celecoxib
NSAIDAnti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
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Cholestyramine
Antihyperlipidemic
Bile acid binding resin (BABR)
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Clofibrate
Antihyperlipidemic
Lipoprotein lipase activator
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Clopidogrel
Antiplatelet
ADP receptor antagonist
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Colchicine
Antigout onlyAnti-inflammatory
Microtubule inhibitor
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Colestipol
Antihyperlipidemic
Bile acid binding resin (BABR)
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Cortisol (Hydrocortisone)
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroid
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Cromolyn sodium
Mast cell stabilizer
Inhibits release ofmast cell mediators
Used prophylactically in asthma
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Dalteparin
Anticoagulant
LMW HeparinATIII activator
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Dexamethasone
AdrenocorticosteroidGlucocorticoidAntineoplastic
Antiemetic
Anti-inflammatory steroidNot by inhalation
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Diflunisal
NSAIDAnalgesic, Anti-inflammatory
Antipyretic
Cyclooxygenase inhibitor
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Dipyridamole
Antiplatelet
Phosphodiesterase inhibitor(increases cAMP)
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Drotrecogin alfa(Activated Protein C)
Anticoagulant
Many actionsTreatment for septic shock
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Enoxaparin
Anticoagulant
LMW HeparinATIII activator
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Eptifibatide
Antiplatelet
GPIIb/IIIa antagonist
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Erythropoietin (EPO)
Cytokine
Primary regulator of RBC synthesis
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Etanercept
TNF inhibitor
Tumor necrosis factor receptor+ Fc portion of IgG
Used in rheumatoid arthritis
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Ezitimibe
Antihyperlipidemic
Cholesterol absorption inhibitor
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Fenofibrate
Antihyperlipidemic
Lipoprotein lipase activator
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Flunisolide
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled
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Fluticasone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled
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Fluvastatin
Antihyperlipidemic
HMG-CoA Reductase Inhibitor
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Gemfibrozil
Antihyperlipidemic
Lipoprotein lipase activator
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Gold salts
Disease modifying anti-rheumatic drugs (DMARD)
auranofin, aurothioglucose
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Granulocyte-Colony Stimulating Factor (G-
CSF)
Cytokine
Granulocyte synthesis stimulator
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Granulocyte/Monocyte-Colony Stimulating Factor
(GM-CSF)
Cytokine
WBC (granulocytes and monocyte) synthesis stimulator
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Heparin
Anticoagulant
ATIII activator
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Hirudin
Anticoagulant
Direct thrombin inhibitor(DTI)
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Histamine
Inflammatory mediator
Stored in mast cells and basophils
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Hydrocortisone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroid
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Hydroxychloroquine
Disease modifyinganti-rheumatic drug (DMARD)
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4-Hydroxycoumarin
Oral anticoagulant
Vitamin K synthesis inhibitor
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Ibuprofen
NSAIDAnalgesic, Anti-inflammatory
Antipyretic
Reversible cyclooxygenase inhibitor
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Indomethacin
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitorTocolytic
Uterine relaxant
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Infliximab
TNF inhibitor
Anti-TNF monoclonal antibodyTreatment of IBD
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Interferon alpha
Antiviral for hepatitisAntineoplastic
Cytokine
Anti-angiogenesis
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Interleukin 2
Cytokine Antineoplastic
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Interleukin 11
Cytokine Antineoplastic (supporting
agent)
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Kallidin
Inflammatory mediator
Plasma, hypotension, pain
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Ketoprofen
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Lepirudin
Anticoagulant
Direct thrombin inhibitor (DTI)
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Leukotriene B4 (LTB4)
Inflammatory mediator
Lipoxygenase productof arachidonate metabolism
Chemotactic
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Leukotrienes C4, D4, E4
(LTC4, LTD4, LTE4)
Inflammatory mediators
Cysteinyl leukotrienesPeptidyl leukotrienes
SRS-ALipoxygenase products ofarachidonate metabolism
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Lovastatin
Antihyperlipidemic
HMG-CoA reductase inhibitor
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Meclofenamate
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Mesalamine(5-ASA)
NSAID (salicylate)
Treatment of IBD
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Methylprednisolone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidNot by inhalation
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Montelukast
Leukotriene inhibitor
LTR1 and LTD4 antagonistAsthma treatment
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Naproxen
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Nedocromil
Mast cell stabilizer
Inhibits release of mast cell mediators
Used prophylactically in asthma
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Nicotinic acid
Antihyperlipidemic
Inhibition of VLDL secretion (?)
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Non-steroidalAnti-inflammatory Drugs
(NSAIDs)
Analgesic, Anti-inflammatory, Antipyretic
Cyclooxygenase inhibitors
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Olsalazine
NSAID (salicylate)
Treatment of IBD
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Phytonadione
Vitamin K
Warfarin antagonist
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Piroxicam
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Platelet Activating Factor (PAF)
Inflammatory mediator
LipidHypotensive
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Pravastatin
Antihyperlipidemic
HMG-CoA reductase inhibitor
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Prednisone
AdrenocorticosteroidGlucocorticoid Antineoplastic
Anti-inflammatoryNot by inhalation
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Probenecid
Uricosuric
Adjunct in penicillin therapy
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Probucol
Antihyperlipidemic
LDL oxidation inhibitor
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Prostaglandin E2 (PGE2)Dinoprostone (Dinoprost)
Oxytocic prostaglandinInflammatory mediator
Cyclooxygenase product of arachidonate metabolism
Uterine stimulantCervical ripener
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Prostaglandin F2 (PGF2)
Inflammatory mediator
Cyclooxygenase product of arachidonate metabolism
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Prostaglandin I2 (PGI2)
Inflammatory mediator
Inhibits platelet aggregation
Cyclooxygenase product of arachidonate metabolism
Prostacyclin
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Protamine Sulfate
Heparin antagonist
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Rofecoxib
NSAIDAnti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
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Simvastatin
Antihyperlipidemic
HMG-CoA reductase inhibitor
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Streptokinase
Thrombolytic
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Rofecoxib
NSAIDAnti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
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Sulfasalazine
Disease modifyinganti-rheumatic drug (DMARD)
Metabolized to sulfonamide+ salicylate (NSAID)
Treatment of IBD
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Sulfinpyrazone
Uricosuric
Anti-gout
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Sulindac
NSAIDAnalgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
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Thrombopoietin
Cytokine
Platelet synthesis stimulator
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Thromboxane A2 (TXA2)
Autacoid
Promotes platelet aggregation Cyclooxygenase product of arachidonate metabolism
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Ticlopidine
Antiplatelet
ADP receptor antagonist
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Tissue plasminogen activators
Thrombolytics
alteplase, reteplase, tenecteplase
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Triamcinolone
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled
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Tumor necrosis factor
CytokineAntineoplastic
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Urokinase
Thrombolytic
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Warfarin
Anticoagulant
Vitamin K synthesis inhibitor
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Zafirlukast
Leukotriene inhibitor
LTR1 and LTD4 antagonistAsthma treatment
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Zileuton
Leukotriene inhibitor
5-lipoxygenase inhibitorUsed in asthma